| Steady-state activation | Steady-state inactivation |  | ||
---|---|---|---|---|---|
 | V1/2-a | Ka | V1/2-i | Ki | n |
Control | −30.0 ± 1.22 | 6.90 ± 0.54 | −71.9 ± 0.90 | 6.97 ± 0.66 | 6 |
BmK I | −42.0 ± 1.31* | 7.05 ± 0.52 | −75.6 ± 1.07 | 10.25 ± 0.64 | 5 |
BmK I-mix | −48.6 ± 1.40** | 3.29 ± 0.49* | −76.8 ± 0.62 | 9.26 ± 0.33 | 5 |
Control | −25.7 ± 1.81 | 4.27 ± 0.59 | −69.2 ± 1.12 | 7.78 ± 0.67 | 6 |
BmK IT2 | −38.1 ± 0.98* | 4.48 ± 0.38 | −72.2 ± 0.86 | 7.91 ± 0.36 | 5 |
BmK IT2-mix | −30.1 ± 1.74 | 5.81 ± 0.73 | −71.6 ± 1.06 | 9.84 ± 0.56 | 5 |